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Ixabiso elifanelekileyo le (R)

Ixabiso elifanelekileyo le (R)

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CAS no: 181289-33-8

Iimpawu zeMichiza: I-Pregabalin Intermediates


Iinkcukacha zeMveliso

Iithegi zeMveliso

Sinenjongo yokuqonda ukonakaliswa komgangatho ekudalweni kunye nokubonelela ngeenkonzo ezifanelekileyo kubathengi basekhaya nabaphesheya ngentliziyo epheleleyo ngexabiso eliQinisekileyo le (R), Samkela abathengi abatsha nabadala abavela kuzo zonke iinkalo zobomi ukuba baqhagamshelane nathi kubudlelwane beshishini elizayo kunye nempumelelo efanayo.
Sinenjongo yokuqonda ukonakaliswa komgangatho ekudalweni kunye nokubonelela ngeenkonzo ezifanelekileyo kubathengi basekhaya nabaphesheya ngentliziyo iphela(-) -3-Carbamoymethyl-5-Methylhexanoic Acid, Nceda uzive ukhululekile ngokunyanisekileyo ukusithumela iimfuno zakho kwaye siya kukuphendula ngokukhawuleza.Sineqela lobunjineli elinamava ukuze likusebenzele malunga nazo zonke iimfuno ezibanzi.Iisampulu ezingahlawulelwayo zinokuthunyelwa ukuze zihambelane neemfuno zakho ukuze uqonde ulwazi oluninzi.Ngomzamo wokuhlangabezana neemfuno zakho, kufuneka uzive ukhululekile ukunxibelelana nathi.Unokusithumelela ii-imeyile kwaye uqhagamshelane nathi ngokuthe ngqo.Ngapha koko, siyakwamkela ukutyelelwa komzi-mveliso wethu osuka kwihlabathi liphela ukuze siqondwe ngcono ngakumbi ngombutho wethu.kunye nezinto.Kurhwebo lwethu nabarhwebi bamazwe amaninzi, sikholisa ukubambelela kumgaqo wolingano kunye nenzuzo efanayo.Ngokwenene lithemba lethu lokuthengisa, ngeenzame ezidibeneyo, urhwebo ngalunye kunye nobuhlobo ukuze sizuze thina.Sijonge phambili ekufumaneni imibuzo yakho.

(R)-(-) -3-Carbamoymethyl-5-methylhexanoic acid isetyenziswa njengendawo ephakathi yePregabalin.
I-Pregabalin ingeyomntu ongeyena i-γ- GABA i-agonist receptor okanye i-antagonist luhlobo olutsha lwe-calcium channel regulator, enokuthintela i-voltage exhomekeke kwi-calcium channels kunye nokunciphisa ukukhululwa kwee-neurotransmitters.Ngokonyango, isetyenziselwa kakhulu i-neuralgia enxulumene nesifo seswekile se-peripheral neuropathy, i-post herpetic neuralgia kunye ne-adjuvant unyango lwabantu abadala abathintekayo, ukuphazamiseka kokukhathazeka ngokubanzi, i-neuralgia ephakathi (kubandakanya i-neuralgia ehambelana nokulimala komgogodla, i-stroke kunye ne-multiple sclerosis) kunye ne-fibromyalgia.

Sinenjongo yokuqonda ukonakaliswa komgangatho ekudalweni kunye nokubonelela ngeenkonzo ezifanelekileyo kubathengi basekhaya nabaphesheya ngentliziyo epheleleyo ngexabiso eliQinisekileyo le (R), Samkela abathengi abatsha nabadala abavela kuzo zonke iinkalo zobomi ukuba baqhagamshelane nathi kubudlelwane beshishini elizayo kunye nempumelelo efanayo.
Ixabiso elifanelekileyo(-) -3-Carbamoymethyl-5-Methylhexanoic Acid, Nceda uzive ukhululekile ngokunyanisekileyo ukusithumela iimfuno zakho kwaye siya kukuphendula ngokukhawuleza.Sineqela lobunjineli elinamava ukuze likusebenzele malunga nazo zonke iimfuno ezibanzi.Iisampulu ezingahlawulelwayo zinokuthunyelwa ukuze zihambelane neemfuno zakho ukuze uqonde ulwazi oluninzi.Ngomzamo wokuhlangabezana neemfuno zakho, kufuneka uzive ukhululekile ukunxibelelana nathi.Unokusithumelela ii-imeyile kwaye uqhagamshelane nathi ngokuthe ngqo.Ngapha koko, siyakwamkela ukutyelelwa komzi-mveliso wethu osuka kwihlabathi liphela ukuze siqondwe ngcono ngakumbi ngombutho wethu.kunye nezinto.Kurhwebo lwethu nabarhwebi bamazwe amaninzi, sikholisa ukubambelela kumgaqo wolingano kunye nenzuzo efanayo.Ngokwenene lithemba lethu lokuthengisa, ngeenzame ezidibeneyo, urhwebo ngalunye kunye nobuhlobo ukuze sizuze thina.Sijonge phambili ekufumaneni imibuzo yakho.


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